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Doxofylline (CAS # 69975-86-6)

Umutungo wa Shimi:

Inzira ya molekulari C11H14N4O4
Misa 266.25
Ubucucike 1.2896 (igereranya)
Ingingo yo gushonga 144-146 ° C.
Ingingo ya Boling 409.46 ° C (igereranya)
Flash point 259.3 ° C.
Amazi meza Gukemura
Gukemura Gushonga mumazi, acetone, Ethyl acetate, benzene, chloroform, dioxane, methanol ishyushye cyangwa Ethanol ishyushye, hafi yo kudashonga muri ether cyangwa peteroli ether.
Umwuka 2.49E-10mmHg kuri 25 ° C.
Kugaragara Crystallisation
Ibara Umweru Kuri Off-White
Merk 14.3438
pKa 0.42 ± 0.70 (Byahanuwe)
Imiterere y'Ububiko munsi ya gaze ya inert (azote cyangwa Argon) kuri 2-8 ° C.
Ironderero 1.6000 (ikigereranyo)
MDL MFCD00865218

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Ibyago n'umutekano

Ibimenyetso bya Hazard Xi - Kurakara
Kode y'ingaruka 36/37/38 - Kurakaza amaso, sisitemu yubuhumekero nuruhu.
Ibisobanuro byumutekano S26 - Mugihe uhuye namaso, kwoza ako kanya n'amazi menshi hanyuma ushakishe inama mubuvuzi.
S36 / 37 - Wambare imyenda ikingira hamwe na gants.
RTECS XH5135000
Kode ya HS 29399990
Uburozi LD50 mu mbeba (mg / kg): 841 mu kanwa; 215.6 iv; mu mbeba: 1022.4 mu kanwa, 445 ip (Franzone)

 

Doxofylline (CAS # 69975-86-6) Kumenyekanisha

Kumenyekanisha Doxofylline (CAS # 69975-86-6) - bronchodilator ya revolution igamije guteza imbere ubuzima bwubuhumekero no kuzamura imibereho yabantu bafite ibibazo byubuhumekero budakira. Nkumunyamuryango wurwego rwimiti ya xanthine, Doxofylline itanga uburyo bwihariye bwibikorwa bitandukanya na bronchodilator gakondo, bikaba byongeweho byingenzi mubikoresho byo kuvura indwara ya asima nindwara zidakira zidakira (COPD).

Doxofylline ikora mu koroshya imitsi yoroshye yumuyaga, biganisha ku guhumeka neza no kugabanya ibibazo byubuhumekero. Ibikorwa byayo byombi ntabwo byagura gusa ibice bya bronchial ahubwo binagira imiti igabanya ubukana, bikemura ikibazo cyo gutwika gikunze kwangiza imyanya y'ubuhumekero. Ibi bituma Doxofylline ihitamo neza kubarwayi bashaka koroherwa no guhumeka, guhumeka neza, nibindi bimenyetso bifitanye isano na asima na COPD.

Kimwe mu bintu bigaragara biranga Doxofylline ni umwirondoro wacyo mwiza. Bitandukanye nabandi ba bronchodilator, ntibishobora gutera ingaruka nka tachycardia cyangwa gastrointestinal guhungabana, bigatuma bikoreshwa mugihe kirekire. Byongeye kandi, Doxofylline iraboneka muburyo butandukanye, harimo ibinini na inhaleri, bitanga uburyo bworoshye kandi bworohereza abarwayi mugucunga imiterere yabo.

Hamwe nibikorwa byiza n'umutekano byagaragaye, Doxofylline ihita ihinduka ihitamo mubashinzwe ubuzima. Iha imbaraga abarwayi kugenzura ubuzima bwabo bwubuhumekero, ibemerera kwishora mubikorwa bya buri munsi bafite ikizere kandi byoroshye.

Inararibonye itandukaniro na Doxofylline - umufasha wizewe mukurwanya indwara zubuhumekero. Baza abashinzwe ubuzima uyu munsi kugirango umenye byinshi byukuntu Doxofylline ishobora kugufasha guhumeka neza no kubaho neza.


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