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ibicuruzwa

H-GLU (OET) -OH (CAS # 1119-33-1)

Umutungo wa Shimi:

Inzira ya molekulari C7H13NO4
Misa 175.18
Ubucucike 1.197g / cm3
Ingingo yo gushonga ~ 179 ° C (Ukuboza)
Ingingo ya Boling 326.5 ° C kuri 760 mmHg
Flash point 151.3 ° C.
Amazi meza Gushonga mumazi 100 mg / ml.
Umwuka 4.29E-05mmHg kuri 25 ° C.
Kugaragara Ifu yishusho, ibara ryera kugeza hanze-yera
pKa 2.21 ± 0.10 (Byahanuwe)
Imiterere y'Ububiko Bika ahantu hijimye, Bifunze byumye, Ubike muri firigo, munsi ya -20 ° C.

Ibicuruzwa birambuye

Ibicuruzwa

Kumenyekanisha H-GLU (OET) -OH (URUBANZA # 1119-33-1), ibice bigezweho bigenda bihindura urwego rwibinyabuzima nubushakashatsi bwa farumasi. Ibicuruzwa bishya nibikomoka kuri acide glutamic, yagenewe kuzamura imbaraga za bioavailable ya miti ivura. Nuburyo bwihariye, H-GLU (OET) -OH itanga urubuga rutandukanye rwo guteza imbere ibiyobyabwenge, rukaba igikoresho cyingenzi kubashakashatsi ndetse nabashinzwe gukora.

H-GLU (OET) -OH irangwa no guhagarara kwayo bidasanzwe no guhuza na sisitemu zitandukanye. Guhindura Ethyl ester ntabwo ihindura gusa ibisubizo mubidukikije byamazi ahubwo binorohereza kwinjizwa muburyo bworoshye. Ibi bituma iba umukandida mwiza kubisabwa muri sisitemu yo gutanga imiti, aho gukoresha neza imiti ikora neza ari ngombwa.

Usibye ibyiza byo gukemuka, H-GLU (OET) -OH yerekana imiti myiza ya farumasi, itanga uburyo bwiza bwo kwinjiza no gukwirakwiza mumubiri. Uru ruganda rufite akamaro kanini mugutezimbere ubuvuzi bwa peptide bushingiye ku buvuzi, aho kuzamura itangwa rya bioactive peptide bishobora kugira ingaruka zikomeye kumusaruro.

Abashakashatsi bazishimira uburyo bworoshye bwo gukoresha no gukoresha H-GLU (OET) -OH, kuko iboneka mu isuku ryinshi kandi irashobora kwinjizwa muri protocole zitandukanye zigerageza. Waba ukora mubuvumbuzi bwibiyobyabwenge, guteza imbere formulaire, cyangwa ubushakashatsi bwamasomo, H-GLU (OET) -OH yiteguye kuba ikirangirire muri laboratoire yawe.

Fungura ubushobozi bwubushakashatsi bwawe hamwe na H-GLU (OET) -OH (CAS #1119-33-1). Inararibonye itandukaniro iyi nterahamwe ishobora gukora mumishinga yawe, kandi utere intambwe mugushakisha ibisubizo byiza kandi byiza byo kuvura. Emera ejo hazaza h'ibinyabuzima hamwe na H-GLU (OET) -OH, aho siyanse ihura nudushya.


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